2. Flavopiridol was the first semi-synthetic cyclin-dependentkinase inhibitor to be tested in clinical trials. Research hasshown that co-administration of flavopiridol with drugs such asthe taxanes had synergistic cytotoxic effects against a variety oftumour cells.HOно.HOCI2.2 Name two classes of compounds that appear in the structureof flavopiridol.

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Answered: 2.2 Name two classes of compounds that…

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Chemistry

2.2 Name two classes of compounds that appear in the structure of flavopiridol.

Organic And Biological Chemistry

7th Edition

ISBN:9781305081079

Author:STOKER, H. Stephen (howard Stephen)

Publisher:STOKER, H. Stephen (howard Stephen)

Chapter9: Proteins

Section: Chapter Questions

Problem 9.58EP

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Question

2. Flavopiridol was the first semi-synthetic cyclin-dependent
kinase inhibitor to be tested in clinical trials. Research has
shown that co-administration of flavopiridol with drugs such as
the taxanes had synergistic cytotoxic effects against a variety of
tumour cells.
HO
но.
HO
CI
2.2 Name two classes of compounds that appear in the structure
of flavopiridol.

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