How does physicochemical properties of a drug define its biological mechanism? Please explain at your own words.

Q: What is pharmacophore? write about its significance in drug discovery? briefly explain

A: The drug is the chemical substance that is responsible for altering the function of living things.…

Q: What is the ultimate goal of drug metabolism? Discuss with example.

A: Drugs are any substances when taken into the body bring out psychological and physiological changes…

Q: Please design a hypothetical targeted drug delivery system and explain it in detail

A: Drug targeting refers to the delivery of medications to specific receptors, organs, or other bodily…

Q: Explain the effect of COM-blockers on bacterial transformation and their application in controlling…

A: Pathogens are disease-causing organisms that can cause humans to become ill or die depending on the…

Q: What is the reason why essential drugs need to be accessilble for all people?

A: WHO defines Essential drugs, as the drugs that satisfy the priority helathcare needs of the people.…

Q: Explain the role of LC50 in ensuring the safety of a drug candidate? Explain at your own words

A: Drugs are defined as the type of chemical substances where they produce changes in the physiology or…

Q: intercalating agent

A: Intercalation is the process in which there is the insertion of molecules between the planar bases…

Q: Define therapeutic index and explain its importance.

A: Therapeutic Index is also known as Therapeutic Ratio. It is a quantitative measurement of the…

Q: Describe the different types of trials a new drug must undergo before it is “ready for market.”

A: A drug is a chemical substance that produces a biological effect. When the drug is taken by…

Q: In what cellular process does the drug target play a role?

A: Cells are separated from their surroundings by the cell membrane.

Q: Lead discovery - Target selection - Medicinal chemistry - In vitro studies - In vivo studies -…

A: THR DRUG DEVELOPMENT PROCESS There are 5 processes of drug development. 1. Drug discovery and…

Q: Explain how different types of reversible inhibitors can be identified.

A: An enzyme inhibitor is a molecule that binds to an enzyme and decreases its activity.

Q: How we can improve pharmacodynamics factors( Receptors) for the development of H1-Antihistamine…

A: First of all, we will know about the terms pharmacodynamics factors (Receptors) and H1 -…

Q: Biotransformation is an important concept in pharmacology, which amongst others,  enables the…

A: Introduction:-  A crucial stage in the cessation of action and removal of therapeutically useful…

Q: explain what scaffold hopping is and why it is useful for drug development?

A: According to the question we have to explain scaffold hopping. In addition to that, we need to…

Q: Describe the influence of protein binding on drug bioavailability

A: Protein binding is the extent to which drugs can bind to proteins in the blood or tissues. The…

Q: Describe the five basic mechanisms of drug resistance.

A: Antibiotics are the drugs which are used to kill the pathogenic bacteria. Penicillin is the first…

Q: The key element that would transform a matrix-type extended-release drug product to a reservoir-type…

A: Answer--  water insoluble rate cintrolling Membrane

Q: List all the possible modes of entry of the drug to the target cell membranes.

A: There are different ways of entry of drugs to the target cell membrane. The most important ones are…

Q: Please What Is the main difference between Medicines and Drugs?

A: A disease is diagnosed based on certain symptoms and laboratory tests. Some diseases require…

Q: What do you know about pharmacodynamic and pharmacokinetic drug development?

A: Drug development begins in the laboratory with lab. and animal testing to ensure complete safety.…

Q: How we can improve (potency, selectivity and decrease in toxicity ) for the development of a…

A: Antihistamines are drugs that are used to treat allergic conditions like sneezing, runny nose,…

Q: Discuss the difference between first-generation and second-generation antihistamines

A: Antihistamines is a family of drug used for the treatment of allergic reactions. Histamines are…

Q: What are the different sources of drugs? Give an example of a drug from each of these sources

A: A drug is a chemical substance which when introduced into a living organism is responsible for…

Q: What is Anti-D Drug?

A: A drug is a substance which is prescribed to treat an infection or disease. It changes the…

Q: Write the Drug Discovery Process of Diltiazem?

A: *The revelation of Ca++ antagonism as a modern principle of activity of coronary drugs comes back to…

Q: Explain the drug discovery process of Losartan?

A: Drug discovery process of Losartan Saralasin is an octa-peptide counterpart of Ang II that replaces…

Q: how does protein binding affect the drug action

A: Many drug molecules interact with the plasma protein and tissue proteins or with other important…

Q: What are Targeted drug delivery systems ? Please explain the ideal properties of Targeted drug…

A: A drug is a molecule which might resemble a organic molecule inside the body or an exogenous…

Q: Choose (+) if the following circumstances or situations will most likely result to production of…

A: Hi! Thank you for the question. We are authorized to answer three to four subparts at a time, since…

Q: Give two examples of macromolecules that are chosen as drug targets.  What are antiseptics? Give an…

A: Macromolecules are the molecules having large molecular mass. These are mostly polymers.

Q: What is the process that leads to drug tolerance?

A: The effect of the drug lessens with repeated exposure. Bigger doses drug is required to bring…

Q: Describe the role of receptor sites in drug action.

A: Receptors are the macromolecule which are present in the membrane or in the cell wall, that…

Q: What are the categories of controlled subtances? What is/are its definition?  Can you please give me…

A: A drug is a substance when administered into a person's body, that causes a change in either the…

Q: Please write the Drug Discovery process  of Losartan?  Please write at your own words.

A: Losartan is a antihypertensive drug which was the first angiotensin II receptor antagonist. The…

Q: Explain how drugs may interact with nucleic acids as a drug target, and outline how a medicinal…

A: Drugs are used to treat a disease. The disease is caused when there is a deviation from the normal.…

Q: What is drug stability in pharmacy?

A: It is asked, what is drug stability in pharmacy?

Q: Briefly discuss how we can improve pharmacodynamic properties of H1-Antihistamine drugs?

A: The study involving the biochemical reactions and effect of the drug on the body is called…

Q: Define the concept of drug bioavailability and briefly explain how it is experimentally determined.…

A: bio-availability of a drug is the indicator or measure to check how much the administered dosage of…

Q: Draw curved arrows to show the mechanism of how TS becomes covalently bound to the drug in its…

A: Trifluridine is an antiviral drug that is used for viral infection in eye. It is used topically and…

Q: What do you know about pharmacodynamic and pharmacokinetic drug development? Explain briefly

A: Drug research:It encompasses many diverse disciplines that are united for a common goal, the…

Q: What are the three main targets of drug design and development?

A: Any non-food substances that bring out changes in psychology and physiology when taken in are called…