2. Which is a false statement regarding non-competitive enzyme inhibitor? (a) It binds to an allosteric site of the enzyme (b) It does not compete with the natural substrate for binding to the active site of the enzy (c) Its binding to the enzyme can induce a conformational change of the enzyme (d) It can be used in combination therapies with a competitive inhibitor (e) It usually is a mimic of the natural enzyme substrate 3. What is the purpose of structure-activity-relationship (SAR) studies? (a) To identify the drug target (b) To improve the pharmacokinetic properties of the drug (c) To determine which atoms or functional groups are important to the activity of a drug (d) To simplify the synthesis of the drug

2. Which is a false statement regarding non-competitive enzyme inhibitor? (a) It binds to an allosteric site of the enzyme (b) It does not compete with the natural substrate for binding to the active site of the enzy (c) Its binding to the enzyme can induce a conformational change of the enzyme (d) It can be used in combination therapies with a competitive inhibitor (e) It usually is a mimic of the natural enzyme substrate 3. What is the purpose of structure-activity-relationship (SAR) studies? (a) To identify the drug target (b) To improve the pharmacokinetic properties of the drug (c) To determine which atoms or functional groups are important to the activity of a drug (d) To simplify the synthesis of the drug

Introductory Chemistry: An Active Learning Approach

6th Edition

ISBN:9781305079250

Author:Mark S. Cracolice, Ed Peters

Publisher:Mark S. Cracolice, Ed Peters

Chapter22: Biochemistry

Section: Chapter Questions

Problem 22.3TC

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Similar questions

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Cytochrome c is an enzyme found in the cells of all aerobic organisms. Elemental analysis of cytochrome c shows that it contains 0.43% iron. What is the minimum molecular weight of this enzyme?
Draw a graph that shows the effect of increasing substrate concentration on the rate of an enzyme-catalyzed reaction (at constant temperature, pH, and enzyme concentration).